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[sixty one] Like lots of other cardiotoxic drugs, methadone blocks the hERG K+ channel. The 2 enantiomers of methadone inhibit hERG channels with various potency. Dextromethadone, which is significantly less powerful as an opioid, is more strong at blocking the hERG channel with an IC50 of ~12 μM. Levomethadone includes a lower affinity, with an I